« Previous
Next »
International Journal of Antimicrobial Agents
Volume 14, Issue 3
, Pages 193-201
, April 2000
Chemistry and biological activity of new 3-benzazepines
References
-
.
The chemistry and pharmacology of 3-benzazepines.
Drugs Future. 1985;10:645–696
- . Narcotic antagonist activity of substituted 1,2,4,5-tetrahydro-3H,3-benzazepines. Narcotic antagonists. In: Braude MC, Harris LS, May EL, Smith JP, Villarreal JE editor. Advances in Biochemical Psychopharmacology. 8:New York: Raven Press; 1974;p. 167–186
-
Cytotoxic activity and radical intensity of 3-benzazopine derivatives.
In:
Chakrabarty AN, Molnár J, Dastidar SG, Motohashi N editor. Non Antibiotics. New Delhi, India: NISCOM; 1998;
-
The effect of some new 3-benzazepines on plasmid DNA, mdr P-glycoprotein and reverse transcriptase leukaemia.
In:
Chakrabarty AN, Molnár J, Dastidar SG, Motohashi N editor. Non Antibiotics. New Delhi, India: NISCOM; 1998;
- Relationship between radical intensity and cytotoxic activity of dopamine-related compounds. Anticancer Res. 1998;18:1069–1074
-
.
Synthesis of benzazepine alkaloids and related compounds.
Heterocycles. 1975;3:931–1004
-
.
Use of the triflamide group for Friedel–Crafts acylation of N-(β-phenethyl)amino acids to 3-benzazepine derivatives.
Heterocycles. 1997;45:1121–1129
-
.
Synthesis of 2-trifluoromethyl-2,3,4,5-tetrahydro-1H-3-benzazepine derivatives.
Heterocycles. 1998;48:555–560
-
Proctor GR, Thomson RH. Azabenzocycloheptenones. Part 1. The Friedel Crafts reaction with aryl-amino-acids, J Chem Soc 1957;2302–2311.
-
.
The Dakin West reaction of N-acyl-1,2,3,4-tetrahydroisoquinoline-1-carboxylic acids using trifluoroacetic anhydride: structural revision for the unexpected product.
Heterocycles. 1998;48:285–294
- . Asymmetric synthesis and reactivities of cis-N-(ρ-toluenesulfinyl)aziridine-2-carboxylic acids. J. Org. Chem. 1994;59:3243–3245
-
.
Apoptosis induced by anticancer drugs.
Cancer Metastasis. 1992;11:121–139
- . Effect of an iron-chelator on ascorbate induced cytotoxicity. Free Radic. Biol. Med. 1997;23:260–270
- . Radical modulation activity of benzo[a]phenothiazine. Anticancer Res. 1997;17:2539–2544
- . Simultaneous determination of uric and ascorbic acids in human serum by reversed-phase high performance liquid chromatography with electrochemical detection. Anal. Biochem. 1984;141:238–243
- . Crystal structure at 3.5 Å resolution of HIV-1 reverse transcriptase complexed with an inhibitor. Science. 1992;256:1783–1790
- . Clinical trials of agents that reverse multidrug resistance. Cancer. 1993;72:3553–3563
-
.
Behavior of N-acylated daunorubicins in mdr1 gene transfected and parental cells.
Biochem. Pharm. 1995;50:889–892
- . The biochemistry of P-glycoprotein-mediated multidrug resistance. Annu. Rev. Biochem. 1989;58:137–171
- . Role of efflux pump(s) in intrinsic resistance of Pseudomonas aeruginosa: active efflux as a contributing factor to β-lactam resistance. Antimicrob. Agents Chemother. 1994;38:1742–1752
- . Correlation between rhodamine 123 accumulation and azole sensitivity in Candida species: possible role for drug efflux in drug resistance. Antimicrob. Agents Chemother. 1996;40:419–425
- . Mycobacterium tuberculosis induces expression of P-gycoprotein in promonocytic U1 cells chronically infected with HIV type 1. Biochem. Biophys. Res. Commun. 1994;199:1181–1187
- . Pharmacology of drugs that alter multidrug resistance in cancer. Pharmacol. Rev. 1990;42:155–199
- . Physical chemical properties shared by compounds that modulate multidrug resistance in human leukemic cells. Mol. Pharmacol. 1988;33:454–462
- . Overcoming of vincristine resistance in P388 leukemia in vivo and in vitro through enhanced cytotoxicity of vincristine and vinblastine by verapamil. Cancer Res. 1981;41:1967–1972
- Structural requirements for activity of propafenone-type modulators in P-glycoprotein-mediated multidrug resistance. Mol. Pharmacol. 1996;49:1122–1130
- Activities of newly synthesized dihydropyridines in overcoming of vincristine resistance, calcium antagonism, and inhibition of photoaffinity labeling of P-glycoprotein in rodents. Cancer Res. 1990;50:310–317
- . Molecular modeling of phenothiazines and related drugs as multidrug resistance modifiers: a comparative molecular field analysis study. J. Med. Chem. 1998;41:1815–1826
- . Cyclosporins as drug resistance modifiers. Biochem. Pharmacol. 1992;43:109–117
- New purines and purine analogs as modulators of multidrug resistance. J. Med. Chem. 1996;39:4099–4108
- . In vitro and in vivo reversal of multidrug resistance by GF120918, an acridonecarboxamide derivative. Cancer Res. 1993;53:4595–4602
- Reversal of mutidrug resistance by a novel quinoline derivative, MS-209. Cancer Chemother. Pharmacol. 1995;35:271–277
- . Total synthesis of stipiamide and designed polyenes as new agents for the reversal of mutidrug resistance. J. Am. Chem. Soc. 1997;119:12159–12169
- . Exploring multidrug resistance using rhodamine 123. Cancer Commun. 1989;1:145–149
- . Studies on the autoxidation of dopamine: interaction with ascorbate. Arch. Biochem. Biophys. 1988;263:447–452
- . Ascorbic acid enhances the cytotoxic effect of 6-hydroxydopamine for human neuroblastoma cell lines. Neurosci. Lett. 1981;26:151–155
- . Ascorbate and phenolic antioxidant interactions in prevention of liposomal oxidation. Lipids. 1992;27:543–550
-
.
Catecholamine analogs as potential antitumor agents.
J. Pharm. Sci. 1979;78:1519–1521
- . Biochemical and toxicological properties of the oxidation products of catecholamines. Free Radic. Biol. Med. 1992;13:391–405
-
Mechanism of antitumoral activity of catechols in culture.
Biochem. Pharm. 1987;36:417–425
-
.
Hospital-acquired infections: diseases with increasingly limited therapies.
Proc. Natl. Acad. Sci. 1994;91:2420–2427
- . Structure activity relationship studies on benzofuran analogs of propafenone-type modulators of tumor cell multidrug resistance. J. Med. Chem. 1996;39:4767–4774
- Novel non-nucleoside inhibitors of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase. 4. 2-Substituted dipyridodiazepinones as potent inhibitors of both wild-type and cysteine-181 HIV-1 reverse. J. Med. Chem. 1995;38:4830–4838
- 5H-Pyrrolo[1,2-b][1,2,5]benzothia-diazepines (PBTDs): a novel class of non-nucleoside reverse transcriptase inhibitors. Bioorg. Med. Chem. 1996;4:837–850
- . Synthesis of a non-nucleoside reverse transcriptase inhibitor in the alkenyidiarylmethane (ADAM) series with optimized potency and therapeutic index. Bioorg. Med. Chem. Lett. 1998;8:195–198
PII: S0924-8579(99)00155-7
© 2000 Elsevier Science B.V. All rights reserved.
« Previous
Next »
International Journal of Antimicrobial Agents
Volume 14, Issue 3
, Pages 193-201
, April 2000
